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Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity
10.1021/acs.jmedchem.7b01670
American Chemical Society
Antoni R. Blaazer
Abhimanyu K. Singh
Erik de Heuvel
Ewald Edink
Kristina M. Orrling
Johan J. N. Veerman
Toine van den Bergh
Chimed Jansen
Erin Balasubramaniam
Wouter J. Mooij
Hans Custers
Maarten Sijm
Daniel N. A. Tagoe
Titilola D. Kalejaiye
Jane C. Munday
Hermann Tenor
An Matheeussen
Maikel Wijtmans
Marco Siderius
Chris de Graaf
Louis Maes
Harry P. de Koning
David S. Bailey
Geert Jan Sterk
Iwan J. P. de Esch
David G. Brown
Rob Leurs
application/pdf
research-article
http://pubs.acs.org/doi/suppl/10.1021/acs.jmedchem.7b01670
© 2018 American Chemical Society
American Chemical Society
True
© 2018 American Chemical Society
© 2018 American Chemical Society
Issue
10.1021/acs.jmedchem.7b01670
VoR
04/19/2018
61
9
3870
3888
© 2018 American Chemical Society
article
0022-2623
1520-4804
Journal of Medicinal Chemistry
research-article
Issue10.1021/acs.jmedchem.7b01670VoR
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