Synthesis of DOTA-conjugated multimeric [Tyr3]octreotide peptides via a combination of Cu(I)-catalyzed "click" cycloaddition and thio acid/sulfonyl azide "sulfo-Click" Amidation and Their in Vivo Evaluation

Yim, C.-B., Dijkgraaf, I., Merkx, R., Versluis, C., Eek, A., Mulder, G.E., Rijkers, D.T.S., Boerman, O.C. and Liskamp, R.M.J. (2010) Synthesis of DOTA-conjugated multimeric [Tyr3]octreotide peptides via a combination of Cu(I)-catalyzed "click" cycloaddition and thio acid/sulfonyl azide "sulfo-Click" Amidation and Their in Vivo Evaluation. Journal of Medicinal Chemistry, 53(10), pp. 3944-3953. (doi:10.1021/jm100246m)

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Item Type:Articles
Status:Published
Refereed:Yes
Glasgow Author(s) Enlighten ID:Liskamp, Professor Robert
Authors: Yim, C.-B., Dijkgraaf, I., Merkx, R., Versluis, C., Eek, A., Mulder, G.E., Rijkers, D.T.S., Boerman, O.C., and Liskamp, R.M.J.
College/School:College of Science and Engineering > School of Chemistry
Journal Name:Journal of Medicinal Chemistry
ISSN:0022-2623
ISSN (Online):1520-4804

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